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- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- GT20029 Experimental topical drug designed to break down androgen receptors
- Fluridil Topical anti-androgen sold as a cosmetic lotion
- Caffeine Stimulant used in hair shampoos and lotions
- RU58841 Experimental topical anti-androgen sold as a research chemical