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- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Fluridil Topical anti-androgen sold as a cosmetic lotion
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride