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- Azelaic Acid Acid used in acne and rosacea creams
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Tretinoin Vitamin A retinoid cream, prescribed for acne
- RU58841 Experimental topical anti-androgen sold as a research chemical
- GT20029 Experimental topical drug designed to break down androgen receptors