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- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- GT20029 Experimental topical drug designed to break down androgen receptors
- HMI-115 Experimental antibody that blocks the prolactin receptor
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug