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- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Metformin Diabetes drug that lowers blood sugar
- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects
- Valproic acid Anti-seizure and mood-stabilising drug
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug