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- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- RU58841 Experimental topical anti-androgen sold as a research chemical
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug