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    Intestinal Permeability Study of Minoxidil: Assessment of Minoxidil as a High Permeability Reference Drug for Biopharmaceutics Classification

    January 2015 in “ Molecular Pharmaceutics ”
    Makoto Ozawa, Yasuhiro Tsume, Moran Zur … Gordon L. Amidon
    Studysummary This study suggests that minoxidil may serve as a suitable reference drug for high permeability classification in the Biopharmaceutics Classification System due to its consistent permeability across different intestinal segments and pH levels.
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    Research cited in this study 4

    1. The Pharmacokinetics of 2.5- to 10-mg Oral Doses of Minoxidil in Healthy Volunteers The Journal of Clinical Pharmacology · 1989
    2. Pharmacology and Pharmacokinetics of Minoxidil Journal of Cardiovascular Pharmacology · 1980
    3. Metabolism of Minoxidil, a New Hypotensive Agent: Biotransformation Following Oral Administration to Rats, Dogs, and Monkeys Journal of Pharmaceutical Sciences · 1975
    4. Pharmacokinetic Studies of Minoxidil Clinical Pharmacology & Therapeutics · 1972

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    2. Intestinal Permeability Study of Minoxidil: Assessment of Minoxidil as a High Permeability Reference Drug for Biopharmaceutics Classification Molecular Pharmaceutics · 2015