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- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- PP405 mitochondrial pyruvate carrier (MPC) inhibitor by Pelage in early trials
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- Rapamycin Immune-suppressing drug, also called sirolimus
- Valproic acid Anti-seizure and mood-stabilising drug