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- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- RU58841 Experimental topical anti-androgen sold as a research chemical
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects
- Lavender Plant essential oil used in scalp products