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- Biotin B vitamin, often sold as a hair supplement
- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- RU58841 Experimental topical anti-androgen sold as a research chemical
- Saw Palmetto Palm-berry extract taken as a supplement