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- Latanoprost Prostaglandin eye drop used for glaucoma
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects