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- PP405 mitochondrial pyruvate carrier (MPC) inhibitor by Pelage in early trials
- Latanoprost Prostaglandin eye drop used for glaucoma
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- RU58841 Experimental topical anti-androgen sold as a research chemical