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- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects
- Valproic acid Anti-seizure and mood-stabilising drug
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug