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- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Caffeine Stimulant used in hair shampoos and lotions
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream