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- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Lavender Plant essential oil used in scalp products
- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor