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- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Caffeine Stimulant used in hair shampoos and lotions
- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor