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- GT20029 Experimental topical drug designed to break down androgen receptors
- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Fluridil Topical anti-androgen sold as a cosmetic lotion
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream