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- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Saw Palmetto Palm-berry extract taken as a supplement