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- GT20029 Experimental topical drug designed to break down androgen receptors
- Fluridil Topical anti-androgen sold as a cosmetic lotion
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Valproic acid Anti-seizure and mood-stabilising drug
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet