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- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- GT20029 Experimental topical drug designed to break down androgen receptors
- Saw Palmetto Palm-berry extract taken as a supplement