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- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Biotin B vitamin, often sold as a hair supplement
- Latanoprost Prostaglandin eye drop used for glaucoma
- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Ketoconazole Antifungal, best known as a dandruff shampoo