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- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Ketoconazole Antifungal, best known as a dandruff shampoo
- Tretinoin Vitamin A retinoid cream, prescribed for acne
- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects