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- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Biotin B vitamin, often sold as a hair supplement
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Saw Palmetto Palm-berry extract taken as a supplement
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor