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- GT20029 Experimental topical drug designed to break down androgen receptors
- Rapamycin Immune-suppressing drug, also called sirolimus
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Tofacitinib JAK inhibitor pill, an immune-system drug
- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically