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- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Rapamycin Immune-suppressing drug, also called sirolimus
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Tofacitinib JAK inhibitor pill, an immune-system drug
- Baricitinib JAK inhibitor pill used for severe alopecia areata