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- Fluridil Topical anti-androgen sold as a cosmetic lotion
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- RU58841 Experimental topical anti-androgen sold as a research chemical
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor