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- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- GT20029 Experimental topical drug designed to break down androgen receptors
- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically