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- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- RU58841 Experimental topical anti-androgen sold as a research chemical
- HMI-115 Experimental antibody that blocks the prolactin receptor
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- GHK-Cu Copper peptide used in skin and hair cosmetics