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- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Metformin Diabetes drug that lowers blood sugar
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- GHK-Cu Copper peptide used in skin and hair cosmetics
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug