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- Fluridil Topical anti-androgen sold as a cosmetic lotion
- HMI-115 Experimental antibody that blocks the prolactin receptor
- Ketoconazole Antifungal, best known as a dandruff shampoo
- Procyanidin Plant polyphenol found in apples and grape seeds
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826