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- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Cetirizine Antihistamine allergy medicine
- Fluridil Topical anti-androgen sold as a cosmetic lotion
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826