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- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Ketoconazole Antifungal, best known as a dandruff shampoo
- Latanoprost Prostaglandin eye drop used for glaucoma