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- GT20029 Experimental topical drug designed to break down androgen receptors
- Stemoxydine Cosmetic ingredient made by L'Oréal
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- Sulforaphane Compound found in broccoli sprouts