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- Fluridil Topical anti-androgen sold as a cosmetic lotion
- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Alfatradiol Weak form of estrogen applied to the scalp
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug