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- Thymosin Beta 4
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- PP405 mitochondrial pyruvate carrier (MPC) inhibitor by Pelage in early trials
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Baricitinib JAK inhibitor pill used for severe alopecia areata