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- Tretinoin Vitamin A retinoid cream, prescribed for acne
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- RU58841 Experimental topical anti-androgen sold as a research chemical