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- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- RU58841 Experimental topical anti-androgen sold as a research chemical
- GT20029 Experimental topical drug designed to break down androgen receptors
- Adenosine Molecule the body uses for energy, used as a cosmetic hair-lotion ingredient