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- HMI-115 Experimental antibody that blocks the prolactin receptor
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Redensyl Cosmetic ingredient blend sold for thinning hair
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- PP405 mitochondrial pyruvate carrier (MPC) inhibitor by Pelage in early trials