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- HMI-115 Experimental antibody that blocks the prolactin receptor
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- GT20029 Experimental topical drug designed to break down androgen receptors
- PP405 mitochondrial pyruvate carrier (MPC) inhibitor by Pelage in early trials
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream