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- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- Baricitinib JAK inhibitor pill used for severe alopecia areata
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826