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- Procyanidin Plant polyphenol found in apples and grape seeds
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Ketoconazole Antifungal, best known as a dandruff shampoo
- Bimatoprost Prostaglandin eye drop used for glaucoma and eyelash growth