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- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Tofacitinib JAK inhibitor pill, an immune-system drug
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- Cetirizine Antihistamine allergy medicine