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- GT20029 Experimental topical drug designed to break down androgen receptors
- HMI-115 Experimental antibody that blocks the prolactin receptor
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- RU58841 Experimental topical anti-androgen sold as a research chemical
- KY19382 Experimental compound that activates hair-growth signals, tested only in animals