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- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug
- Verteporfin Light-activated eye drug being studied for scarring
- Rapamycin Immune-suppressing drug, also called sirolimus
- Estradiol Estrogen hormone, prescribed in tablet, patch and gel forms