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- Estradiol Estrogen hormone, prescribed in tablet, patch and gel forms
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Thymosin Beta 4
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826