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- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Baricitinib JAK inhibitor pill used for severe alopecia areata
- PP405 mitochondrial pyruvate carrier (MPC) inhibitor by Pelage in early trials
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet