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- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- RU58841 Experimental topical anti-androgen sold as a research chemical
- Bicalutamide Nonsteroidal anti-androgen, originally a prostate cancer drug