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- Dutasteride 5-alpha reductase inhibitor that blocks both enzyme types, a stronger DHT blocker than finasteride
- Minoxidil Vasodilator used on the scalp and, at low doses, as a tablet
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Saw Palmetto Palm-berry extract taken as a supplement
- Melatonin Hormone that regulates sleep, sold as a supplement