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- Finasteride Popular 5-alpha reductase inhibitor that lowers DHT, taken as a pill or used topically
- Neem Oil Oil from the neem tree, used in traditional remedies
- Cyproterone a synthetic anti-androgen and weak progestogen that inhibits DHT binding to androgen receptor
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Fluridil Topical anti-androgen sold as a cosmetic lotion