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- Procyanidin Plant polyphenol found in apples and grape seeds
- Pyrilutamide Experimental topical anti-androgen, also known as KX-826
- Clascoterone Topical androgen-receptor blocker, approved as an acne cream
- Stemoxydine Cosmetic ingredient made by L'Oréal
- Spironolactone Blood-pressure and diuretic drug with anti-androgen effects